Appendix Table A.

Primary Care to Relevant Potentially Inappropriate Medications from Beers Criteria*

Therapeutic Category/DrugRecommendationTherapeutic Category/DrugRecommendation
Anticholinergics (Excludes TCAs)AvoidBarbituratesAvoid
    Brompheniramine (oral)    Butalbital
    Carbinoxamine    Phenobarbital
    ChlorpheniramineBenzodiazepinesAvoid for treatment of insomnia, agitation, or delirium
    Clemastine    Short and interm. acting
    Cyproheptadine        Alprazolam
    Dexbrompheniramine        Estazolam
    Dexchlorpheniramine        Lorazepam
    Diphenhydramine        Oxazepam
    Doxylamine        Temazepam
    Hydroxyzine        Triazolam
    Promethazine    Long acting
    Triprolidine        Chlorazepate
Antiparkinson agents        Chlordiazepoxide
    BenztropineAvoid        Chlordiazepoxide-amitriptyline
    Trihexyphenidyl        Clidinium-chlordiazepoxide
AntispasmodicsAvoid except in short-term palliative care        Clonazepam
    Belladonna alkaloids        Diazepam
    Clidinium-chlordiazepoxide        Flurazepam
    Dicyclomine        Quazepam
    HyoscyamineNonbenzodiazepine hypnoticsAvoid chronic use (>90 days)
    Propantheline    Eszopiclone
    Scopolamine    Zolpidem
Tertiary TCAs (Alone or in Combination)Avoid    Zaleplon
    AmitriptylineMegestrolAvoid
    Chlordiazepoxide-amitriptylineMeprobamateAvoid
    ClomipramineTrimethobenzamideAvoid
    ImipraminePain Medications
    Perphenazine-amitriptyline    MeperidineAvoid
    Trimipramine    IndomethacinAvoid
ThioridazineAvoid    Ketorolac (oral)Avoid
MesoridazineAvoidSkeletal muscle relaxantsAvoid
Dessicated thyroidAvoid    Carisoprodol
TestosteroneAvoid unless indicated for moderate to severe hypogonadism    Chlorzoxazone
    Cyclobenzaprine
    Metaxalone
Estrogens with/without progestinsAvoid oral and topical patch    Methocarbamol
    Orphenadrine
Sulfonylureas, long durationAvoid
    Chlorpropamide
    Glyburide
  • TCA, tricyclic antidepressant.

  • * Primary care–relevant PIMs were selected from Table 2 of 2012 American Geriatric Society Beers Criteria for Potentially Inappropriate Medication Use in Older Adults.24